The asymmetric synthesis of α,α’-dibenzyl esters 1 from α-benzyl acrylates and diversely substituted boronic acids was performed by Christopher Frost and co-workers from University of Bath (Org. 1345728-51-9 Formula Lett.…
Stephen Caddick and co-workers from University College London were successful in the generation of peptidomimetics via stereoselectivecross-metathesis (Org. Biomol. Chem. Formula of 37342-97-5 2007, 5, ASAP.DOI: 10.1039/b700804j). By applying Grubbs’…
G resolution; T2 time point at which the maximum transform of F340/F380 was reached soon after the substitution of the SBS with the NH4Cl bathing remedy; T3 time point (at…
By about 1.5 whereas for homooligomeric BAX the improvement is about four Additionally, making use of of SDSL-EPR distance data mitigates theJ Struct Biol. Author manuscript; obtainable in PMC 2017…
The groups of Fernando Cossio from Universidad del País Vasco-Euskal Herriko Unibertsitatea and Angel Díaz-Ortiz from Universidad de Castilla-La Mancha, Spain, have made investigations toward the stereochemical outcome for the…
The group of Lal Dhar Yadav from the University of Allahabad, India, has reported on a Biginelli-type reaction of unprotected aldoses, 2-methyl-2-phenyl-1,3-oxathiolan-5-one 1 as CH-acidic building block and urea/thiourea under…
Hydrozirconation is a mild method for the selective preparation of functionalized organometallics and its compatibility with a range of common protecting groups represents a considerable advantage of these species over…
Diastereoselectivity in ring-closing metathesis can be achieved under either kinetic or thermodynamic control. PMID:23539298 Siegfried Blechert of the Technische Universität Berlin has found (Angew. Chem. Int. Ed. 2006, 45, 1302.…
The group of Samuel Danishefsky from Columbia University has reported on an oxidative dearomatization/transannular Diels-Alder sequence as key step in the total synthesis of (±)-11-O-debenzoyltashironin (4) (J. Am. Chem. Soc.…
Erin DiMauro and Joseph Kennedy from Amgen have developed a microwave protocol for the synthesis of a focused library of 3-amino-imidazopyridines 3 (J. Org. Chem. 2007, 72, 1013. DOI: 10.1021/jo0622072).…
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